Mu opioid receptor antagonist 2 [CAS 2773925-64-5]
Mu opioid receptor antagonist 2 [CAS 2773925-64-5]
SKU:QM-0065885
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Product Details
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Description
Mu opioid receptor antagonist 2 (compound 25) is a potent, selective and blood-brain barrier (BBB) penetrant μ opioid receptor (MOR) antagonist with a Ki of 0.37 nM and an EC50 of 0.44 nM. Mu opioid receptor antagonist 2 has remarkable CNS antagonism against morphine, and precipitated fewer withdrawal symptoms than Naloxone. Mu opioid receptor antagonist 2 can be used for researching opioid use disorders (OUD) [1].
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CAS Number
[2773925-64-5]
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Molecular Formula
C25H28N2O4S
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Molecular Weight
452.57
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Smiles
O[C@]12[C@H]3CC4=C5[C@@]1(CCN3CC6CC6)[C@H]([C@H](CC2)NC(C7=CC=CS7)=O)OC5=C(O)C=C4
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Target
Opioid Receptor
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Isoform
μ Opioid Receptor/MOR
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Mu opioid receptor antagonist 2 [CAS 2773925-64-5]
Mu opioid receptor antagonist 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.