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NR1H4 activator 1 [CAS 2242855-68-9]
NR1H4 activator 1 [CAS 2242855-68-9]
SKU:QM-0060779
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Product Details
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Description
NR1H4 activator 1 is a potent and selective Famesoid X Receptor (FXR) agonist, extracted from patent WO2018152171A1, example 4. NR1H4 activator 1 shows strong FXR agonistic potency with a EC50 value of 1 nM in a Human FXR (NR1H4) Assay. NR1H4 activator 1 has the potential for treatment of gastrointestinal disease[1].
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CAS Number
[2242855-68-9]
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Molecular Formula
C34H53NO7S
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Molecular Weight
619.85
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Smiles
C[C@@]12[C@@H]([C@H](C)COC(NS(=O)(C3=CC=C(OC(C)C)C=C3)=O)=O)CC[C@@]1([H])[C@]4([H])[C@H](O)[C@H](CC)[C@]5([H])C[C@@H](O)CC[C@]5(C)[C@@]4([H])CC2
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Target
FXR
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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NR1H4 activator 1 [CAS 2242855-68-9]
NR1H4 activator 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.