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NR2B-selective NMDA receptor antagonist 1 [CAS 457897-92-6]
NR2B-selective NMDA receptor antagonist 1 [CAS 457897-92-6]
SKU:QM-0101000-01
£122.88 GBP
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Product Details
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Description
NR2B-selective NMDA receptor antagonist 1 (compound 29) is a potent antagonist of NR1/NR2B receptors, with IC50s of 0.05 μM, 0.73 μM, 2.4 μM to NR1/NR2B NMDA receptor, hERG, α1-AdR, respectivity. NR2B-selective NMDA receptor antagonist 1 exhibites efficient permeability across the blood–brain barrier[1].
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CAS Number
[457897-92-6]
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Molecular Formula
C18H22Cl2N2O4S
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Molecular Weight
433.35
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Smiles
CS(NC1=CC=C(C=C1)OC[C@@H](O)CNCCC2=CC(Cl)=C(C=C2)Cl)(=O)=O
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Target
IGluR; Potassium Channel
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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NR2B-selective NMDA receptor antagonist 1 [CAS 457897-92-6]
NR2B-selective NMDA receptor antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.