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NSD2-PWWP1 ligand 1
NSD2-PWWP1 ligand 1
SKU:QM-0109047
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Product Details
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Description
NSD2-PWWP1 ligand 1 (compound 34) is a small molecule ligand targeting the NSD2-PWWP1 domain (pIC50: 8.2) . NSD2 is a large multidomain protein with histone writer and histone reader functions. Dysregulation of the levels of histone methyltransferase nuclear receptor binding SET domain 2 (NSD2) may lead to a variety of hematological and solid malignancies. NSD2-PWWP1 ligand 1 binds to NSD2, reducing its enzymatic activity and inhibiting tumorigenesis[1].
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Molecular Formula
C25H27N3O3
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Molecular Weight
417.5
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Smiles
CC1=CC=C(C=C1C2=NOC(C)=C2C3=CC4=C(NC(CO4)=O)C=C3)CN5CCCCC5
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Target
Histone Methyltransferase
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Shipping Conditions
Room temperature
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NSD2-PWWP1 ligand 1
NSD2-PWWP1 ligand 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.