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PAR2 modulator-1 [CAS 2378159-28-3]
PAR2 modulator-1 [CAS 2378159-28-3]
SKU:QM-0009804
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Product Details
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Description
PAR2 modulator-1 (Compound C781) is a protease activated receptor type 2 (PAR2) antagonist. PAR2 modulator-1 can specifically inhibit the PAR2-dependent MAPK signaling pathway with an IC50 value of 8.5 μM. PAR2 modulator-1 can block the pain response triggered by PAR2 agonists. PAR2 modulator-1 can be used for the researches of inflammation, immunology and neurological disease, such as chronic pain and asthma[1].
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CAS Number
[2378159-28-3]
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Molecular Formula
C27H41N5O5
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Molecular Weight
515.64
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Smiles
O=C(C1=CC=CO1)N2C3([H])N(C([C@@H](C2)NC(CC(C)C)=O)=O)[C@@H](C(N(C3)CC4CCNCC4)=O)CC(C)C
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Target
P38 MAPK; Protease Activated Receptor (PAR)
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Shipping Conditions
Room temperature
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PAR2 modulator-1 [CAS 2378159-28-3]
PAR2 modulator-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.