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PAR4 antagonist 2
PAR4 antagonist 2
SKU:QM-0085060
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Product Details
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Description
PAR4 antagonist 2 (Compound 31) is a protease activated receptor 4 (PAR4) antagonist, with IC50 values of 95 nM and 367 nM for human PAR4 and mouse PAR4. PAR4 antagonist 2 is active against PAR4 activation by the native protease thrombin cleavage but not the synthetic PAR4 agonist peptide AYPGKF[1].
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Molecular Formula
C22H18F2N6O
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Molecular Weight
420.41
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Smiles
O=C(NC1=NNC(C2=C(F)C=C(F)C=C2)=N1)C3=NN(C4=CC=CC=C4)C5=C3CCCC5
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Target
Protease Activated Receptor (PAR)
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Isoform
PAR4
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PAR4 antagonist 2
PAR4 antagonist 2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.