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PAR4 antagonist 3 [CAS 3057206-40-0]
PAR4 antagonist 3 [CAS 3057206-40-0]
SKU:QM-0101731
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Product Details
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Description
PAR4 antagonist 3 (Compound 36) is a selective antagonist for protease activated receptor 4 (PAR4) . PAR4 antagonist 3 exhibits antiplatelet efficacy with IC50 of 26.1 nM. PAR4 antagonist 3 improves metabolic stablility in human liver microsomes with T1/2 of 97.6 min[1].
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CAS Number
[3057206-40-0]
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Molecular Formula
C22H16FN3O5S
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Molecular Weight
453.44
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Smiles
FC1=CC=C(OCC2COC3=CC=C4C(OC(C5=CN6C(SC(OC)=N6)=N5)=C4)=C3O2)C=C1
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Target
Protease Activated Receptor (PAR)
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Isoform
PAR4
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PAR4 antagonist 3 [CAS 3057206-40-0]
PAR4 antagonist 3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.