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PI3K/mTOR Inhibitor-1 [CAS 1949802-49-6]
PI3K/mTOR Inhibitor-1 [CAS 1949802-49-6]
SKU:QM-0058548
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Product Details
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Description
PI3K/mTOR Inhibitor-1 is a potent, orally bioavailable dual PI3K/mTOR inhibitor with IC50s of 20/376/204/46 nM and 186 nM for PI3Kα/PI3Kβ/PI3Kγ/PI3Kδ and mTOR, respectively[1]. Antitumor activity[1].
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CAS Number
[1949802-49-6]
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Molecular Formula
C18H22FN5O3S
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Molecular Weight
407.46
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Smiles
NC1=CC(F)=C(C2=CC(C3(CC3)S(=O)(C)=O)=NC(N4[C@@H](C)COCC4)=N2)C=N1
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Target
MTOR; PI3K
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Isoform
MTOR; PI3Kα; PI3Kβ; PI3Kγ; PI3Kδ
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PI3K/mTOR Inhibitor-1 [CAS 1949802-49-6]
PI3K/mTOR Inhibitor-1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.