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PPARγ/δ modulator 1 [CAS 2089159-00-0]
PPARγ/δ modulator 1 [CAS 2089159-00-0]
SKU:QM-0067547
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Product Details
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Description
PPARγ/δ modulator 1 (compound 3e) is a potent PPAR modulator. PPARγ/δ modulator 1 is a PPARδ antagonist and a PPARγ partial agonist , with Ki values of 14.4 nM and 5.31 μM, respectively. PPARγ/δ modulator 1 has the EC50 of 7.3 and 12.6 μM for PPARδ corepression and adiponectin production, respectively[1].
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CAS Number
[2089159-00-0]
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Molecular Formula
C18H18ClIN6O3Se
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Molecular Weight
607.69
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Smiles
O[C@H]1[C@H]([C@@H]([Se][C@@H]1C(NC)=O)N2C3=C(N=C2)C(NCC4=CC=CC(I)=C4)=NC(Cl)=N3)O
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Target
PPAR
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Isoform
PPARγ; PPARδ
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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PPARγ/δ modulator 1 [CAS 2089159-00-0]
PPARγ/δ modulator 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.