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Progranulin modulator-2

Progranulin modulator-2

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SKU:QM-0119579

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  • Description

    Progranulin modulator-2 (compound 18A) is a bromodomain and extra-terminal domain (BET) inhibitor. Progranulin modulator-2 enhances PGRN expression by targeting members of the BET protein family. Progranulin modulator-2 can be used to study the role of BET protein in neurodevelopment, neuroplasticity and neurodegeneration[1].

  • Molecular Formula

    C19H14FN3O2

  • Molecular Weight

    335.33

  • Smiles

    O=C1C(NC=C2)=C2C(C3=CC=CN=C3OC4=CC=C(F)C=C4)=CN1C

  • Target

    Epigenetic Reader Domain

  • Shipping Conditions

    Room temperature

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Progranulin modulator-2

Progranulin modulator-2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.