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PROTAC ERRα ligand 1 [CAS 1264754-13-3]

PROTAC ERRα ligand 1 [CAS 1264754-13-3]

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QM-0077209-01

£200.66 GBP
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Product Details

  • Description

    PROTAC ERRα ligand 1 is a PROTAC target protein ligand. PROTAC ERRα ligand 1 is an orally active ERRα inverse agonist with IC50 values of 0.6 μM for ERRα. PROTAC ERRα ligand 1 shows no significant activity against a panel of other nuclear receptors, including ERαc, ERRγ, ERβ, PPARα, PPARγ, PPARδ, and RXRα. PROTAC ERRα ligand 1 can provide enhanced insulin sensitivity in vivo. PROTAC ERRα ligand 1 can be used for metabolic diseases research, such as type 2 diabetes and obesity[1].

  • CAS Number

    [1264754-13-3]

  • Molecular Formula

    C19H11F3N2O4S

  • Molecular Weight

    420.36

  • Smiles

    N#CC1=CC=C(OC2=CC=C(/C=C(SC(N3)=O)/C3=O)C=C2OC)C(C(F)(F)F)=C1

  • Target

    Estrogen Receptor/ERR; Ligands for Target Protein for PROTAC

  • Isoform

    ERRα

  • Purity

    99.47

  • Solubility

    DMSO : 100 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302-H312-H332

  • Precautions

    P261-P264-P270-P271-P280-P302+P352-P304+P340-P330-P363-P501
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Variant Variant total Quantity Price Variant total
5 mgQM-0077209-01
5 mgQM-0077209-01
£200.66/ea		 £0.00
£200.66/ea £0.00
10 mgQM-0077209-02
10 mgQM-0077209-02
£275.99/ea		 £0.00
£275.99/ea £0.00
50 mgQM-0077209-03
50 mgQM-0077209-03
£702.46/ea		 £0.00
£702.46/ea £0.00
100 mgQM-0077209-04
100 mgQM-0077209-04
£1,179.95/ea		 £0.00
£1,179.95/ea £0.00
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PROTAC ERRα ligand 1 [CAS 1264754-13-3]

PROTAC ERRα ligand 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.