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Protease-Activated Receptor-1 antagonist 3
Protease-Activated Receptor-1 antagonist 3
SKU:QM-0065238
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Product Details
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Description
Protease-Activated Receptor-1 antagonist 3 is a potent protease-activated receptor-1 antagonist with an IC50 value of 7 nM. Protease-Activated Receptor-1 antagonist 3 shows binding affinity for hERG K+ channel with an IC50 value of 9 μM[1].
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Molecular Formula
C30H34N4O3
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Molecular Weight
498.62
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Smiles
[H][C@]12[C@H]([C@@H]([C@@H](C)[C@H]3[C@]1(C(O[C@@H]2C)=O)CN(C(NCC)=O)C3)C)/C=C/C4=CC=C(C=N4)C5=CC=CC=C5C#N
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Target
Protease Activated Receptor (PAR)
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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Protease-Activated Receptor-1 antagonist 3
Protease-Activated Receptor-1 antagonist 3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.