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Sigma-1 receptor antagonist 3 [CAS 1639220-17-9]

Sigma-1 receptor antagonist 3 [CAS 1639220-17-9]

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SKU:QM-0141619-01

£351.32 GBP
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  • Description

    Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (σ1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 μM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1].

  • CAS Number

    [1639220-17-9]

  • Molecular Formula

    C19H23ClFN3O

  • Molecular Weight

    363.86

  • Smiles

    CC1=NC(C2=CC=C(F)C=C2)=NC(OCCCN3CCCCC3)=C1Cl

  • Target

    Potassium Channel; Sigma Receptor

  • Isoform

    Sigma 1 Receptor

  • Purity

    99.47

  • Solubility

    DMSO : 12.5 mg/mL (ultrasonic)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

  • Hazard Statement

    H302-H315-H319

  • Precautions

    P264-P270-P280-P302+P352-P305+P351+P338-P330-P362+P364-P501

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Variant Variant total Quantity Price Variant total
5 mgQM-0141619-01
5 mgQM-0141619-01
£351.32/ea
£0.00
£351.32/ea £0.00
10 mM - 1 mLQM-0141619-02
10 mM - 1 mLQM-0141619-02
£381.69/ea
£0.00
£381.69/ea £0.00
10 mgQM-0141619-03
10 mgQM-0141619-03
£539.64/ea
£0.00
£539.64/ea £0.00
25 mgQM-0141619-04
25 mgQM-0141619-04
£853.12/ea
£0.00
£853.12/ea £0.00
50 mgQM-0141619-05
50 mgQM-0141619-05
£1,142.29/ea
£0.00
£1,142.29/ea £0.00
100 mgQM-0141619-06
100 mgQM-0141619-06
£1,493.42/ea
£0.00
£1,493.42/ea £0.00

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Sigma-1 receptor antagonist 3 [CAS 1639220-17-9]

Sigma-1 receptor antagonist 3 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.