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TRPC antagonist 1 [CAS 3027139-12-1]
TRPC antagonist 1 [CAS 3027139-12-1]
SKU:QM-0073463
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Product Details
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Description
TRPC antagonist 1 (compound 15g) is a potent TRP channel (TRPC) antagonist with IC50s of 2.4 μM, 12.2 μM, 7.6 μM, 2.9 μM, and 3.4 μM for TRPC3, TRPC4, TRPC5, TPRC6, and TRPC7, respectively. TRPC antagonist 1 displays noteworthy anti-glioblastoma efficacy in vitro against U87 cell lines[1].
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CAS Number
[3027139-12-1]
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Molecular Formula
C23H22N4O2S
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Molecular Weight
418.51
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Smiles
NCCN(C1=NC(C(NC2=CC=C(O)C=C2)=O)=CS1)CC3=CC=C(C=CC=C4)C4=C3
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Target
TRP Channel
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Isoform
TRPC3; TRPC4; TRPC5; TRPC6; TRPC7
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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TRPC antagonist 1 [CAS 3027139-12-1]
TRPC antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.