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TRPV1 antagonist 6
TRPV1 antagonist 6
SKU:QM-0097982
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Product Details
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Description
TRPV1 antagonist 6 (compound 51) is a mode-selective antagonist for transient receptor potential vanilloid member 1 (TRPV1), which shows antagonism with IC50 of 2.85 nM to capsaicin activation and 28.48 % inhibition against proton activation at a 3 µM concentration[1].
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Molecular Formula
C26H28ClN5O3
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Molecular Weight
493.99
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Smiles
CC(C)(C)C1=NN(C(CNC(NC2=CC=CC(N3CCO)=C2C=CC3=O)=O)=C1)C4=CC=CC(Cl)=C4
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Target
TRP Channel
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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TRPV1 antagonist 6
TRPV1 antagonist 6 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.