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TRPV1 antagonist 9 [CAS 939040-79-6]
TRPV1 antagonist 9 [CAS 939040-79-6]
SKU:QM-0119839-01
£911.43 GBP
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Product Details
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Description
TRPV1 antagonist 9 (compound 13c) is an orally active transient receptor potential vanilloid 1 (TRPV1) channel antagonist. TRPV1 antagonist 9 blocks Ca2+ uptake by CHO cells expressing TRPV1 receptors with IC50 values are 0.6 and 0.8 nM for Capsaicin and acid-induced Ca2+ uptake, respectively. TRPV1 antagonist 9 blocks Capsaicin (HY-10448) -induced flinch response and causes hyperthermia in rats[1].
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CAS Number
[939040-79-6]
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Molecular Formula
C22H19F3N6O3
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Molecular Weight
472.42
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Smiles
NC1=NC(C(NC1=O)=CC=C2)=C2OC3=NC(NCCOC)=NC(C4=CC=C(C(F)(F)F)C=C4)=C3
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Target
TRP Channel
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Shipping Conditions
Room temperature
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TRPV1 antagonist 9 [CAS 939040-79-6]
TRPV1 antagonist 9 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.