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V1a/V2 antagonist 1
V1a/V2 antagonist 1
SKU:QM-0089515
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Product Details
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Description
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual V1a and V2 receptor antagonist with high binding affinity for both receptors (Ki: 0.13 nM for hV1a, 0.53 nM for hV2 and 0.5 nM for mV1a; IC50: 2.2 nM for hV1a). V1a/V2 antagonist 1 inhibits Oxytocin -induced scratching behavior in mice[1].
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Molecular Formula
C25H26ClN5O3
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Molecular Weight
479.96
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Smiles
ClC1=CC=C2N3C(N(CC4)CCN4C5=C(OCC6)C6=CC=C5)=NN=C3CC7(OCCO7)CC2=C1
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Target
Vasopressin Receptor
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Isoform
V1a Receptor ; V2 Receptor
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Shipping Conditions
Room temperature
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V1a/V2 antagonist 1
V1a/V2 antagonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.