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VDR agonist 1 [CAS 2269494-43-9]
VDR agonist 1 [CAS 2269494-43-9]
SKU:QM-0058905
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Product Details
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Description
VDR agonist 1 (compound 28) is a nonsteroidal Vitamin D receptor (VDR) agonist, with an IC50 of 690 nM in MCF-7 cells. VDR agonist 1 arrests the cell cycle through the up-regulation of p21 and p27, promotes apoptosis by increasing the expression of BAX and decrease the expression of Bcl-2[1].
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CAS Number
[2269494-43-9]
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Molecular Formula
C32H51N3O2
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Molecular Weight
509.77
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Smiles
O=C(C1=CC(C(CC)(C2=CC=C(/C=C/C(O)(CC)CC)C(C)=C2)CC)=CN1CC)NCCN(CC)CC
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Target
Apoptosis; VD/VDR
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Solubility
10 mM in DMSO
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Shipping Conditions
Room temperature
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VDR agonist 1 [CAS 2269494-43-9]
VDR agonist 1 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.