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VHL Ligand 38 [CAS 1360616-29-0]
VHL Ligand 38 [CAS 1360616-29-0]
SKU:QM-0004854
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Product Details
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Description
VHL Ligand 38 (Compound 1) is a competitive E3 ubiquitin-protein ligase VHL inhibitor with IC50s of 4.1 and 7.0 μM in 1% and 10% DMSO, respectively. VHL Ligand 38 contains a hydroxyproline residue and an isoxazolylacetamide fragment. VHL Ligand 38 significantly inhibits the binding of a fluorescent peptide derived from HIF1α (FAM-DEALA-Hyp-YIPD) to VHL[1].
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CAS Number
[1360616-29-0]
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Molecular Formula
C21H22N4O5
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Molecular Weight
410.42
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Smiles
O=C([C@H]1N(C(CC2=CC(C)=NO2)=O)C[C@H](O)C1)NCC3=CC=C(C4=CN=CO4)C=C3
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Target
E1/E2/E3 Enzyme
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Shipping Conditions
Room temperature
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VHL Ligand 38 [CAS 1360616-29-0]
VHL Ligand 38 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.