Collection: Bioactive Small Molecules
Explore QuantiMol's extensive range of bioactive small molecules for life science research, pathway studies, high-throughput screening, and drug discovery applications. This collection spans the full spectrum of pharmacological activity — including enzyme inhibitors, kinase inhibitors, protease inhibitors, receptor agonists and antagonists, ion channel modulators, epigenetic probes, and signalling pathway tool compounds — covering virtually every major biological target class relevant to modern biomedical research.
Each bioactive small molecule supplied by QuantiMol is rigorously characterised for purity, identity, and biological activity, giving researchers the confidence to use them as primary pharmacological tools in mechanistic studies, target validation, and lead optimisation workflows. Whether you are dissecting a signalling cascade, profiling off-target effects, or building a focused screening library, QuantiMol's bioactive small molecules provide the chemical precision your research demands.
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TLR7 agonist 24
SKU: QM-0089986 | Size: 1 Each Price on request -
TLR7 agonist 12 [CAS 2389988-47-8]
CAS: 2389988-47-8 | SKU: QM-0071044 | Size: 1 Each Price on request -
Thrombin inhibitor 7 [CAS 2866508-00-9]
CAS: 2866508-00-9 | SKU: QM-0069845 | Size: 1 Each Price on request -
Tie2 kinase inhibitor 3 [CAS 870225-11-9]
CAS: 870225-11-9 | SKU: QM-0087613 | Size: 1 Each Price on request -
THR-β agonist 6 [CAS 2791290-58-7]
CAS: 2791290-58-7 | SKU: QM-0068197 | Size: 1 Each Price on request -
TLR8 agonist 2 (hydrochloride) [CAS 2412937-65-4]
CAS: 2412937-65-4 | SKU: QM-0064821 | Size: 1 Each Price on request -
Thyroid hormone receptor beta agonist-1 [CAS 2140902-80-1]
CAS: 2140902-80-1 | SKU: QM-0070627 | Size: 1 Each Price on request -
TLR8 agonist 2 [CAS 2412937-64-3]
CAS: 2412937-64-3 | SKU: QM-0064820 | Size: 1 Each Price on request -
Thrombin inhibitor 6 [CAS 1628224-94-1]
CAS: 1628224-94-1 | SKU: QM-0069770 | Size: 1 Each Price on request -
STING agonist-49-PAB-Ala-Val-CO-C2-mal [CAS 2803608-03-7]
CAS: 2803608-03-7 | SKU: QM-0016205 | Size: 1 Each Price on request -
STING agonist-49-β-D-Glu-benzylalcohol-di (amide-C2) -mal [CAS 2803608-01-5]
CAS: 2803608-01-5 | SKU: QM-0016204 | Size: 1 Each Price on request -
STING agonist-49-CO-C2-mal-Cys [CAS 2803608-05-9]
CAS: 2803608-05-9 | SKU: QM-0016178 | Size: 1 Each Price on request -
STING agonist-49-CO-C2-mal [CAS 2803607-99-8]
CAS: 2803607-99-8 | SKU: QM-0016177 | Size: 1 Each Price on request -
STING agonist-49 [CAS 2138299-66-6]
CAS: 2138299-66-6 | SKU: QM-0016176 | Size: 1 Each Price on request -
STING agonist-48 [CAS 3027712-31-5]
CAS: 3027712-31-5 | SKU: QM-0015612 | Size: 1 Each Price on request -
STING agonist-47
SKU: QM-0015159 | Size: 1 Each Price on request -
STING agonist-45 [CAS 2361424-97-5]
CAS: 2361424-97-5 | SKU: QM-0014480 | Size: 1 Each Price on request -
TAF1 ligand 1 [CAS 1926986-25-5]
CAS: 1926986-25-5 | SKU: QM-0013928 | Size: 1 Each Price on request -
TBK1 ligand 2-C-O-C4-O-C3-O-C-amide [CAS 2052306-12-2]
CAS: 2052306-12-2 | SKU: QM-0013820 | Size: 1 Each Price on request -
TBK1 ligand 2 [CAS 2052306-16-6]
CAS: 2052306-16-6 | SKU: QM-0013819 | Size: 1 Each Price on request -
STING agonist-44
SKU: QM-0013755 | Size: 1 Each Price on request -
STING ligand-4
SKU: QM-0013677 | Size: 1 Each Price on request -
STING agonist-42 [CAS 2942231-48-1]
CAS: 2942231-48-1 | SKU: QM-0013624 | Size: 1 Each Price on request -
TFAM activator 1 [CAS 932992-44-4]
CAS: 932992-44-4 | SKU: QM-0013384-01 | Size: 5 mg£206.74 GBP -
STING agonist-46 [CAS 3033532-05-4]
CAS: 3033532-05-4 | SKU: QM-0013361 | Size: 1 Each Price on request -
TERT ligand-1 [CAS 2412120-47-7]
CAS: 2412120-47-7 | SKU: QM-0011919 | Size: 1 Each Price on request -
TAAR1/5-H-2CR agonist-1 [CAS 3024777-79-2]
CAS: 3024777-79-2 | SKU: QM-0011535 | Size: 1 Each Price on request -
Tau ligand-1 [CAS 3063166-64-0]
CAS: 3063166-64-0 | SKU: QM-0011391 | Size: 1 Each Price on request -
STING agonist-43 [CAS 2882097-31-4]
CAS: 2882097-31-4 | SKU: QM-0010829 | Size: 1 Each Price on request -
TACC3 inhibitor 2 [CAS 2642351-96-8]
CAS: 2642351-96-8 | SKU: QM-0009743 | Size: 1 Each Price on request -
TERT activator-2 [CAS 332939-29-4]
CAS: 332939-29-4 | SKU: QM-0008884-01 | Size: 25 mg£216.46 GBP -
TGR5 Receptor Agonist (Standard) [CAS 1197300-24-5]
CAS: 1197300-24-5 | SKU: QM-0006956-01 | Size: 1 mg£205.52 GBP -
TGF-βRI inhibitor 3 [CAS 666729-57-3]
CAS: 666729-57-3 | SKU: QM-0006580-01 | Size: 5 mg£238.32 GBP -
TDP1 Inhibitor-1 [CAS 2248702-80-7]
CAS: 2248702-80-7 | SKU: QM-0139594-01 | Size: 5 mg£614.98 GBP -
TGR5 Receptor Agonist 4 [CAS 1872436-42-4]
CAS: 1872436-42-4 | SKU: QM-0152142-01 | Size: 5 mg£608.90 GBP -
Syk Inhibitor II [CAS 726695-51-8]
CAS: 726695-51-8 | SKU: QM-0137480-01 | Size: 5 mg£118.38 GBP -
STING agonist-26 [CAS 2868261-48-5]
CAS: 2868261-48-5 | SKU: QM-0150938-01 | Size: 5 mg£912.65 GBP -
TbPTR1 inhibitor 2 [CAS 17557-67-4]
CAS: 17557-67-4 | SKU: QM-0205790-01 | Size: 1 g£51.91 GBP -
TCS PrP Inhibitor 13 [CAS 34320-83-7]
CAS: 34320-83-7 | SKU: QM-0112673-01 | Size: 5 mg£135.25 GBP -
Thalidomide-NH-CBP/p300 ligand 2 [CAS 2484739-21-9]
CAS: 2484739-21-9 | SKU: QM-0146847-01 | Size: 1 mg£649.00 GBP -
STING agonist-7 [CAS 2767442-46-4]
CAS: 2767442-46-4 | SKU: QM-0148022-01 | Size: 5 mg£426.65 GBP -
Succinate/succinate receptor antagonist 1 [CAS 2361972-29-2]
CAS: 2361972-29-2 | SKU: QM-0150249-01 | Size: 5 mg£140.88 GBP -
STING ligand-1 [CAS 2365039-41-2]
CAS: 2365039-41-2 | SKU: QM-0138422-01 | Size: 5 mg£803.30 GBP -
STING agonist-8 (dihydrochloride)
SKU: QM-0148184-01 | Size: 1 mg£614.98 GBP -
STING antagonist-2 [CAS 2305940-34-3]
CAS: 2305940-34-3 | SKU: QM-0149790-01 | Size: 5 mg£1,368.28 GBP -
TAS2R14 agonist-2 [CAS 2883007-69-8]
CAS: 2883007-69-8 | SKU: QM-0151085-01 | Size: 5 mg£357.39 GBP -
TGR5 Receptor Agonist [CAS 1197300-24-5]
CAS: 1197300-24-5 | SKU: QM-0147760-01 | Size: 5 mg£139.75 GBP -
TFEB activator 1 [CAS 39777-61-2]
CAS: 39777-61-2 | SKU: QM-0145232-01 | Size: 5 mg£108.25 GBP -
TDP1 Inhibitor-2 [CAS 859142-95-3]
CAS: 859142-95-3 | SKU: QM-0149449-01 | Size: 5 mg£834.89 GBP -
STING agonist-4 [CAS 2138300-40-8]
CAS: 2138300-40-8 | SKU: QM-0141015-01 | Size: 1 mg£301.50 GBP -
TERT activator-1 [CAS 666699-46-3]
CAS: 666699-46-3 | SKU: QM-0156091-01 | Size: 5 mg£194.59 GBP -
TAO Kinase inhibitor 1 [CAS 850467-66-2]
CAS: 850467-66-2 | SKU: QM-0137356-01 | Size: 5 mg£118.38 GBP -
STING ligand-3 [CAS 2762552-73-6]
CAS: 2762552-73-6 | SKU: QM-0156322-01 | Size: 5 mg£307.58 GBP -
TAK1/MAP4K2 inhibitor 1 [CAS 1315330-11-0]
CAS: 1315330-11-0 | SKU: QM-0077319-01 | Size: 5 mg£514.13 GBP -
STING agonist-3 [CAS 2138299-29-1]
CAS: 2138299-29-1 | SKU: QM-0083459-01 | Size: 5 mg£551.80 GBP -
TFEB activator 2 [CAS 3027414-04-3]
CAS: 3027414-04-3 | SKU: QM-0153217-01 | Size: 5 mg£426.65 GBP -
STING antagonist-1 [CAS 3036981-21-9]
CAS: 3036981-21-9 | SKU: QM-0153412-01 | Size: 5 mg£407.21 GBP -
STING agonist-3 (trihydrochloride)
SKU: QM-0083460-01 | Size: 5 mg£551.80 GBP -
STING agonist-30 [CAS 2951078-67-2]
CAS: 2951078-67-2 | SKU: QM-0150005-01 | Size: 1 mg£621.05 GBP -
TAO Kinase inhibitor 2 [CAS 850467-77-5]
CAS: 850467-77-5 | SKU: QM-0151280-01 | Size: 5 mg£124.00 GBP -
TAAR1 agonist 2 [CAS 1804128-38-8]
CAS: 1804128-38-8 | SKU: QM-0168292 | Size: 1 Each Price on request -
Sulfane sulfur probe 4 [CAS 1810731-98-6]
CAS: 1810731-98-6 | SKU: QM-0152637 | Size: 1 mg£527.50 GBP -
TbPTR1 inhibitor 1 [CAS 2499713-65-2]
CAS: 2499713-65-2 | SKU: QM-0067710 | Size: 1 Each Price on request -
Syk Inhibitor II (dihydrochloride dihydrate) [CAS 1965323-05-0]
CAS: 1965323-05-0 | SKU: QM-0058496 | Size: 1 Each Price on request -
STING agonist-29 [CAS 2868261-51-0]
CAS: 2868261-51-0 | SKU: QM-0070438 | Size: 1 Each Price on request -
TAMRA-probe 1
SKU: QM-0062752 | Size: 1 Each Price on request -
TAS2R14 agonist-1 [CAS 2439115-08-7]
CAS: 2439115-08-7 | SKU: QM-0070554 | Size: 1 Each Price on request -
TAAR1 agonist 1
SKU: QM-0127954 | Size: 1 Each Price on request -
STING agonist-24 [CAS 2408722-91-6]
CAS: 2408722-91-6 | SKU: QM-0070434 | Size: 1 Each Price on request -
TEAD ligand 1 [CAS 2971850-47-0]
CAS: 2971850-47-0 | SKU: QM-0127401 | Size: 1 Each Price on request -
STING agonist-38 [CAS 2850251-27-1]
CAS: 2850251-27-1 | SKU: QM-0126861 | Size: 1 mg£401.13 GBP -
STING agonist-9 [CAS 2653337-73-4]
CAS: 2653337-73-4 | SKU: QM-0067614 | Size: 1 Each Price on request -
STING modulator-5 [CAS 2305940-22-9]
CAS: 2305940-22-9 | SKU: QM-0067982 | Size: 1 Each Price on request -
TAAR1 agonist 1 (hydrochloride)
SKU: QM-0125278 | Size: 1 Each Price on request -
TGR5 agonist 5
SKU: QM-0124279 | Size: 1 Each Price on request -
TGR5 agonist 7
SKU: QM-0119416 | Size: 1 Each Price on request -
TACC3 inhibitor 1 [CAS 3033646-06-6]
CAS: 3033646-06-6 | SKU: QM-0069772 | Size: 1 Each Price on request -
STING modulator-7 [CAS 702662-64-4]
CAS: 702662-64-4 | SKU: QM-0117740-01 | Size: 1 mg£319.73 GBP -
TGR5 Receptor Agonist 3 [CAS 2643391-08-4]
CAS: 2643391-08-4 | SKU: QM-0066884 | Size: 1 Each Price on request -
TAT-PAK18 inhibitory peptide
SKU: QM-0115609 | Size: 1 Each Price on request -
STING agonist-34 [CAS 2913152-30-2]
CAS: 2913152-30-2 | SKU: QM-0068598-01 | Size: 1 mg£499.55 GBP -
STING agonist-31 [CAS 2719001-44-0]
CAS: 2719001-44-0 | SKU: QM-0070679 | Size: 1 Each Price on request -
TAAR1 agonist 3 [CAS 1804129-70-1]
CAS: 1804129-70-1 | SKU: QM-0109447 | Size: 1 Each Price on request -
STING agonist-28 [CAS 2868261-50-9]
CAS: 2868261-50-9 | SKU: QM-0070437 | Size: 1 Each Price on request -
STING agonist-25 [CAS 2408723-10-2]
CAS: 2408723-10-2 | SKU: QM-0070435 | Size: 1 Each Price on request -
T-Type calcium channel inhibitor 2 [CAS 2771965-57-0]
CAS: 2771965-57-0 | SKU: QM-0067501 | Size: 1 Each Price on request -
STING modulator-3 [CAS 2839639-94-8]
CAS: 2839639-94-8 | SKU: QM-0067979 | Size: 1 Each Price on request -
Target Protein Ligand-Linker Conjugates 2
SKU: QM-0105381 | Size: 1 Each Price on request -
TGF-βRI inhibitor 2 [CAS 476474-11-0]
CAS: 476474-11-0 | SKU: QM-0104884-01 | Size: 5 mg£100.38 GBP -
Telomeric G4s ligand 1 [CAS 3047091-81-3]
CAS: 3047091-81-3 | SKU: QM-0104141 | Size: 1 Each Price on request -
TGR5 agonist 6 [CAS 2925211-47-6]
CAS: 2925211-47-6 | SKU: QM-0099411 | Size: 1 Each Price on request -
TGR5 agonist 1
SKU: QM-0068605 | Size: 1 Each Price on request -
TGR5 agonist 2
SKU: QM-0068606 | Size: 1 Each Price on request -
Syncytial Virus Inhibitor-1 [CAS 1422496-79-4]
CAS: 1422496-79-4 | SKU: QM-0059648 | Size: 1 Each Price on request -
STING agonist-27 [CAS 2868261-45-2]
CAS: 2868261-45-2 | SKU: QM-0070436 | Size: 1 Each Price on request -
Syk Inhibitor II (dihydrochloride) [CAS 227449-73-2]
CAS: 227449-73-2 | SKU: QM-0058495 | Size: 1 Each Price on request -
Substance P Receptor Antagonist 1 [CAS 225526-17-0]
CAS: 225526-17-0 | SKU: QM-0001560-01 | Size: 1 mg£972.18 GBP -
TGR5 agonist 4
SKU: QM-0071703 | Size: 1 Each Price on request -
Syk Inhibitor II (hydrochloride) [CAS 2490508-82-0]
CAS: 2490508-82-0 | SKU: QM-0092709 | Size: 1 Each Price on request -
STING agonist-8 [CAS 2745723-90-2]
CAS: 2745723-90-2 | SKU: QM-0065702 | Size: 1 Each Price on request -
TBL1X ligand 1 [CAS 1083160-12-6]
CAS: 1083160-12-6 | SKU: QM-0091576 | Size: 1 Each Price on request -
TGR5 agonist 3 [CAS 2148317-51-3]
CAS: 2148317-51-3 | SKU: QM-0071702 | Size: 1 Each Price on request -
TG2 inhibitor VA4 [CAS 2088001-23-2]
CAS: 2088001-23-2 | SKU: QM-0089754-01 | Size: 5 mg£218.88 GBP -
STING ligand-2 [CAS 1307526-16-4]
CAS: 1307526-16-4 | SKU: QM-0089390 | Size: 1 Each Price on request -
STING agonist-23 [CAS 2361570-16-1]
CAS: 2361570-16-1 | SKU: QM-0070433-01 | Size: 5 mg£583.38 GBP -
STING agonist-33 [CAS 2591300-32-0]
CAS: 2591300-32-0 | SKU: QM-0070861 | Size: 1 Each Price on request -
STING modulator-4 [CAS 2839639-72-2]
CAS: 2839639-72-2 | SKU: QM-0067983 | Size: 1 Each Price on request -
TDP1 Inhibitor-3 [CAS 3074962-67-4]
CAS: 3074962-67-4 | SKU: QM-0078857-01 | Size: 5 mg£375.62 GBP -
TFEB activator 3 [CAS 3027413-48-2]
CAS: 3027413-48-2 | SKU: QM-0078157-01 | Size: 5 mg£301.50 GBP -
SNAP-fusion protein ligand-1 [CAS 913817-45-5]
CAS: 913817-45-5 | SKU: QM-0050892-01 | Size: 100 mg£188.51 GBP -
SSTR4 agonist 6 [CAS 2744188-17-6]
CAS: 2744188-17-6 | SKU: QM-0050572 | Size: 1 Each Price on request -
SMR efflux inhibitor
SKU: QM-0025094 | Size: 1 Each Price on request -
STAT6 ligand-2
SKU: QM-0016378 | Size: 1 Each Price on request -
SSTR3 agonist-1 (TFA)
SKU: QM-0014535 | Size: 1 Each Price on request -
SSTR3 Agonist-1 [CAS 3086695-73-7]
CAS: 3086695-73-7 | SKU: QM-0014534-01 | Size: 1 mg£551.80 GBP -
SST1 receptor antagonist-2 [CAS 524743-70-2]
CAS: 524743-70-2 | SKU: QM-0014440 | Size: 1 Each Price on request -
SST1 receptor antagonist-1 [CAS 868057-23-2]
CAS: 868057-23-2 | SKU: QM-0014437 | Size: 1 Each Price on request -
SMARCA2 Ligand-Linker Conjugate-4 [CAS 3033001-29-2]
CAS: 3033001-29-2 | SKU: QM-0014210 | Size: 1 Each Price on request -
STAT6 ligand-1
SKU: QM-0014202 | Size: 1 Each Price on request -
SMARCA2/4 Ligand-Linker Conjugate 2 [CAS 2380272-29-5]
CAS: 2380272-29-5 | SKU: QM-0014137 | Size: 1 Each Price on request