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PLK1/BRD4-IN-2 [CAS 2251709-89-2]

PLK1/BRD4-IN-2 [CAS 2251709-89-2]

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SKU:QM-0152987-01

£514.13 GBP
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  • Description

    PLK1/BRD4-IN-2 (compound 15) is a BI-2536 analog and dual inhibitor that targets both Polo-like kinase 1 (PLK1) and BRD4bromodomain (BRD4-BD1 IC50=28 nM, PLK1 IC50=40 nM).

  • CAS Number

    [2251709-89-2]

  • Molecular Formula

    C27H36N6O3

  • Molecular Weight

    492.61

  • Smiles

    C[C@H]1N(C2CCCC2)C3=NC(NC4=C(C=C(C=C4)C(N5CCCCCC5)=O)OC)=NC=C3N(C1=O)C

  • Target

    Epigenetic Reader Domain

  • Isoform

    BRD4

  • Purity

    98.92

  • Solubility

    10 mM in DMSO|DMSO : 10 mg/mL (ultrasonic; warming; heat to 60°C)

  • Storage Conditions

    -20°C, 3 years; 4°C, 2 years (Powder)

  • Shipping Conditions

    Room Temperature

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Variant Variant total Quantity Price Variant total
1 mgQM-0152987-01
1 mgQM-0152987-01
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£343.80
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£514.13/ea
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£343.80
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5 mgQM-0152987-02
5 mgQM-0152987-02
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£837.00
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£1,179.95/ea
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£837.00
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£1,179.95/ea
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10 mM - 1 mLQM-0152987-03
10 mM - 1 mLQM-0152987-03
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£906.30
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£1,273.51/ea
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£906.30
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10 mgQM-0152987-04
10 mgQM-0152987-04
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£1,088.10
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£1,518.93/ea
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£1,088.10
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25 mgQM-0152987-05
25 mgQM-0152987-05
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£1,740.60
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£2,399.81/ea
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£1,740.60
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50 mgQM-0152987-06
50 mgQM-0152987-06
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£2,263.50
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£3,105.72/ea
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£2,263.50
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£3,105.72/ea
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100 mgQM-0152987-07
100 mgQM-0152987-07
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£2,942.10
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£4,021.84/ea
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£2,942.10
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£4,021.84/ea
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PLK1/BRD4-IN-2 [CAS 2251709-89-2]

PLK1/BRD4-IN-2 is a premium-grade research compound supplied by Quantimol for laboratory and scientific applications.