Collection: Bioactive Small Molecules
Explore QuantiMol's extensive range of bioactive small molecules for life science research, pathway studies, high-throughput screening, and drug discovery applications. This collection spans the full spectrum of pharmacological activity — including enzyme inhibitors, kinase inhibitors, protease inhibitors, receptor agonists and antagonists, ion channel modulators, epigenetic probes, and signalling pathway tool compounds — covering virtually every major biological target class relevant to modern biomedical research.
Each bioactive small molecule supplied by QuantiMol is rigorously characterised for purity, identity, and biological activity, giving researchers the confidence to use them as primary pharmacological tools in mechanistic studies, target validation, and lead optimisation workflows. Whether you are dissecting a signalling cascade, profiling off-target effects, or building a focused screening library, QuantiMol's bioactive small molecules provide the chemical precision your research demands.
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URAT1 inhibitor 3 [CAS 2850331-30-3]
CAS: 2850331-30-3 | SKU: QM-0150524-01 | Size: 5 mg£351.32 GBP -
Wnt/β-catenin agonist 1 [CAS 2305372-67-0]
CAS: 2305372-67-0 | SKU: QM-0138376-01 | Size: 5 mg£614.98 GBP -
UCK2 Inhibitor-1 [CAS 902289-98-9]
CAS: 902289-98-9 | SKU: QM-0149677-01 | Size: 5 mg£325.81 GBP -
Wnt/β-catenin agonist 2 [CAS 943820-93-7]
CAS: 943820-93-7 | SKU: QM-0147662-01 | Size: 5 mg£301.50 GBP -
Wnt pathway activator 2 [CAS 1360540-82-4]
CAS: 1360540-82-4 | SKU: QM-0145351-01 | Size: 5 mg£206.74 GBP -
YAP/TAZ inhibitor-1 [CAS 2093565-23-0]
CAS: 2093565-23-0 | SKU: QM-0137056-01 | Size: 1 mg£351.32 GBP -
VCP Activator 1 [CAS 3061959-30-3]
CAS: 3061959-30-3 | SKU: QM-0152312-01 | Size: 5 mg£702.46 GBP -
WRN inhibitor 3 [CAS 2923009-48-5]
CAS: 2923009-48-5 | SKU: QM-0152028-01 | Size: 5 mg£607.68 GBP -
URAT1 inhibitor 6 [CAS 2244807-49-4]
CAS: 2244807-49-4 | SKU: QM-0151374-01 | Size: 5 mg£608.90 GBP -
URAT1 inhibitor 8 [CAS 1632005-33-4]
CAS: 1632005-33-4 | SKU: QM-0076078-01 | Size: 5 mg£313.65 GBP -
VHL Ligand 8 [CAS 2701565-76-4]
CAS: 2701565-76-4 | SKU: QM-0144286-01 | Size: 5 mg£246.83 GBP -
VHL Ligand 14 [CAS 2010986-87-3]
CAS: 2010986-87-3 | SKU: QM-0076501-01 | Size: 1 mg£438.80 GBP -
WRN inhibitor 1 [CAS 2923008-44-8]
CAS: 2923008-44-8 | SKU: QM-0151252-01 | Size: 1 mg£1,430.24 GBP -
WT-TTR inhibitor 1 [CAS 23983-05-3]
CAS: 23983-05-3 | SKU: QM-0151204-01 | Size: 5 mg£118.38 GBP -
USP30 inhibitor 11 [CAS 2067332-64-1]
CAS: 2067332-64-1 | SKU: QM-0137158-01 | Size: 1 mg£376.83 GBP -
Y1 receptor antagonist 1 (formic)
SKU: QM-0081483-01 | Size: 5 mg£551.80 GBP -
WRN inhibitor 4 [CAS 2923009-45-2]
CAS: 2923009-45-2 | SKU: QM-0152030-01 | Size: 1 mg£753.49 GBP -
URAT1&XO inhibitor 1 [CAS 2669726-78-5]
CAS: 2669726-78-5 | SKU: QM-0151373-01 | Size: 5 mg£597.97 GBP -
Wnt/β-catenin agonist 3 (hydrochloride)
SKU: QM-0149523-01 | Size: 5 mg£124.00 GBP -
Viability/Cytotoxicity Assay Kit for Live & Dead Cells (Calcein/PI)
SKU: QM-0161806-01 | Size: 500 Tests£110.50 GBP -
Utrophin activator-1 [CAS 381208-40-8]
CAS: 381208-40-8 | SKU: QM-0177395-01 | Size: 1 mg£587.03 GBP -
Wnt pathway inhibitor 3 [CAS 663213-98-7]
CAS: 663213-98-7 | SKU: QM-0151278-01 | Size: 5 mg£78.82 GBP -
URAT1 inhibitor 11 [CAS 2416416-13-0]
CAS: 2416416-13-0 | SKU: QM-0154213 | Size: 1 Each Price on request -
Viral 2C protein inhibitor 1 [CAS 1594427-18-5]
CAS: 1594427-18-5 | SKU: QM-0066702 | Size: 1 Each Price on request -
WRN inhibitor 12 [CAS 3044040-29-8]
CAS: 3044040-29-8 | SKU: QM-0135203 | Size: 1 Each Price on request -
XIAP BIR2/BIR2-3 inhibitor-1 [CAS 1609384-59-9]
CAS: 1609384-59-9 | SKU: QM-0073081 | Size: 1 Each Price on request -
URAT1 inhibitor 5 [CAS 2102670-94-8]
CAS: 2102670-94-8 | SKU: QM-0070742 | Size: 1 Each Price on request -
WRN inhibitor 14
SKU: QM-0133336 | Size: 1 Each Price on request -
URAT1 inhibitor 9 [CAS 2251727-90-7]
CAS: 2251727-90-7 | SKU: QM-0073212 | Size: 1 Each Price on request -
UCK2 Inhibitor-3 [CAS 2376687-49-7]
CAS: 2376687-49-7 | SKU: QM-0067918-01 | Size: 5 mg£678.15 GBP -
Y4R agonist-1 [CAS 2757328-51-9]
CAS: 2757328-51-9 | SKU: QM-0131095 | Size: 1 Each Price on request -
Utrophin modulator 1 [CAS 3068935-32-7]
CAS: 3068935-32-7 | SKU: QM-0068798 | Size: 1 Each Price on request -
UCK2 Inhibitor-2 [CAS 866842-71-9]
CAS: 866842-71-9 | SKU: QM-0067917-01 | Size: 1 mg£1,561.46 GBP -
XIAP/cIAP1 antagonist-1 [CAS 1403898-55-4]
CAS: 1403898-55-4 | SKU: QM-0057195 | Size: 1 Each Price on request -
WRN inhibitor 18 [CAS 3064599-42-1]
CAS: 3064599-42-1 | SKU: QM-0123367 | Size: 1 Each Price on request -
VHL Ligand intermediate-2 [CAS 2380273-24-3]
CAS: 2380273-24-3 | SKU: QM-0074375 | Size: 1 Each Price on request -
URAT1 inhibitor 2 [CAS 2803951-18-8]
CAS: 2803951-18-8 | SKU: QM-0065566 | Size: 1 Each Price on request -
URAT1 inhibitor 4 [CAS 2700292-02-8]
CAS: 2700292-02-8 | SKU: QM-0069789 | Size: 1 Each Price on request -
WRN inhibitor 6
SKU: QM-0119968 | Size: 1 Each Price on request -
VHL Ligand intermediate-1 [CAS 2380273-21-0]
CAS: 2380273-21-0 | SKU: QM-0074374 | Size: 1 Each Price on request -
Vif-ElonginC interaction inhibitor 1 [CAS 374679-27-3]
CAS: 374679-27-3 | SKU: QM-0059787 | Size: 1 Each Price on request -
WRN inhibitor 17 [CAS 3064599-40-9]
CAS: 3064599-40-9 | SKU: QM-0109520 | Size: 1 Each Price on request -
WDR5-MLL1 antagonist 1 [CAS 1422389-91-0]
CAS: 1422389-91-0 | SKU: QM-0109169-01 | Size: 1 mg£262.63 GBP -
WRN inhibitor 10
SKU: QM-0108359 | Size: 1 Each Price on request -
WRN inhibitor 2 [CAS 2923009-56-5]
CAS: 2923009-56-5 | SKU: QM-0070855 | Size: 5 mg£815.45 GBP -
Y4R agonist-2 [CAS 2757328-63-3]
CAS: 2757328-63-3 | SKU: QM-0107640 | Size: 1 Each Price on request -
Y1R probe-1 [CAS 2773476-41-6]
CAS: 2773476-41-6 | SKU: QM-0066399 | Size: 1 Each Price on request -
USP7/USP47 inhibitor 1 [CAS 90680-28-7]
CAS: 90680-28-7 | SKU: QM-0106153-01 | Size: 1 mg£537.21 GBP -
VHL Ligand-Linker Conjugates 15 [CAS 2375564-62-6]
CAS: 2375564-62-6 | SKU: QM-0060760 | Size: 1 Each Price on request -
URAT1 inhibitor 10 [CAS 3012586-38-5]
CAS: 3012586-38-5 | SKU: QM-0104360 | Size: 1 Each Price on request -
WRN inhibitor 15
SKU: QM-0103197 | Size: 1 Each Price on request -
VHL Ligand-Linker Conjugates 17
SKU: QM-0062088 | Size: 1 Each Price on request -
Y1 receptor antagonist 1 [CAS 221697-09-2]
CAS: 221697-09-2 | SKU: QM-0000166 | Size: 1 mg£1,192.10 GBP -
Vasopressin V2 receptor antagonist 2
SKU: QM-0101157-01 | Size: 5 mg£269.91 GBP -
Urinary Trypsin Inhibitor Fragment [CAS 164859-77-2]
CAS: 164859-77-2 | SKU: QM-0100416 | Size: 1 Each Price on request -
USP3 ZnF-UBD ligand-1 [CAS 2419322-41-9]
CAS: 2419322-41-9 | SKU: QM-0072935-01 | Size: 5 mg£426.65 GBP -
WRN inhibitor 11 [CAS 3058317-61-3]
CAS: 3058317-61-3 | SKU: QM-0097410 | Size: 1 Each Price on request -
WRN inhibitor 7 [CAS 444780-45-4]
CAS: 444780-45-4 | SKU: QM-0096296 | Size: 1 Each Price on request -
URAT1 inhibitor 7 [CAS 1632002-28-8]
CAS: 1632002-28-8 | SKU: QM-0070854-01 | Size: 1 mg£499.55 GBP -
XIAP BIR2/BIR2-3 inhibitor-3 [CAS 1434125-52-6]
CAS: 1434125-52-6 | SKU: QM-0073088 | Size: 1 Each Price on request -
Vasopressin V2 receptor antagonist 1 [CAS 2648650-50-2]
CAS: 2648650-50-2 | SKU: QM-0066737 | Size: 1 Each Price on request -
VDR agonist 1 [CAS 2269494-43-9]
CAS: 2269494-43-9 | SKU: QM-0058905 | Size: 1 Each Price on request -
URAT1&XO inhibitor 3 [CAS 2089040-93-5]
CAS: 2089040-93-5 | SKU: QM-0092067 | Size: 1 Each Price on request -
V1a/V2 antagonist 1
SKU: QM-0089515 | Size: 1 Each Price on request -
VDR agonist 2 [CAS 3052323-55-1]
CAS: 3052323-55-1 | SKU: QM-0068681 | Size: 1 Each Price on request -
Wnt pathway inhibitor 4 [CAS 663214-57-1]
CAS: 663214-57-1 | SKU: QM-0070761 | Size: 10 mg£78.82 GBP -
VCP/p97 inhibitor-1 [CAS 2630950-38-6]
CAS: 2630950-38-6 | SKU: QM-0063745-01 | Size: 1 mg£678.15 GBP -
VHL Ligand 8-PEG2-O-piperidine-Boc
SKU: QM-0082405 | Size: 1 Each Price on request -
XIAP antagonist 1 [CAS 375835-04-4]
CAS: 375835-04-4 | SKU: QM-0072804 | Size: 1 Each Price on request -
TRPV4 antagonist 5 [CAS 3026084-12-5]
CAS: 3026084-12-5 | SKU: QM-0016452 | Size: 1 Each Price on request -
TRPV4-KCa2.3 modulator 1 [CAS 2616611-60-8]
CAS: 2616611-60-8 | SKU: QM-0015279 | Size: 1 Each Price on request -
TRPV1 antagonist 11 [CAS 3084843-71-7]
CAS: 3084843-71-7 | SKU: QM-0013583 | Size: 1 Each Price on request -
Tyrosinase activator-1
SKU: QM-0013421 | Size: 1 Each Price on request -
TRPV1 agonist-1 [CAS 2763372-26-3]
CAS: 2763372-26-3 | SKU: QM-0011911 | Size: 1 Each Price on request -
Type II TRK inhibitor 3
SKU: QM-0011774 | Size: 1 Each Price on request -
TYK2 ligand 2 [CAS 2924460-80-8]
CAS: 2924460-80-8 | SKU: QM-0011453 | Size: 1 Each Price on request -
TRPV1 antagonist 10 [CAS 896584-55-7]
CAS: 896584-55-7 | SKU: QM-0010941 | Size: 1 Each Price on request -
Tubulin inhibitor 50
SKU: QM-0010796 | Size: 1 Each Price on request -
TYK2 activator-1 [CAS 3087219-47-1]
CAS: 3087219-47-1 | SKU: QM-0010777 | Size: 1 Each Price on request -
TSPO/Carbonic Anhydrase Modulator 1
SKU: QM-0009124 | Size: 1 Each Price on request -
Tubulin inhibitor 49 (hydrobromide)
SKU: QM-0009087-01 | Size: 5 mg£218.88 GBP -
Tubulin inhibitor 49 [CAS 1023875-75-3]
CAS: 1023875-75-3 | SKU: QM-0009086-01 | Size: 5 mg£218.88 GBP -
Ubiquitin Isopeptidase Inhibitor I, G5 (Standard) [CAS 108477-18-5]
CAS: 108477-18-5 | SKU: QM-0002007 | Size: 1 Each Price on request -
TSHR antagonist S37a [CAS 2143452-20-2]
CAS: 2143452-20-2 | SKU: QM-0143016-01 | Size: 5 mg£627.13 GBP -
Tubulin inhibitor 11 [CAS 2366260-33-3]
CAS: 2366260-33-3 | SKU: QM-0150762-01 | Size: 5 mg£238.32 GBP -
Tubulin inhibitor 1 [CAS 2237054-53-2]
CAS: 2237054-53-2 | SKU: QM-0137585-01 | Size: 5 mg£118.38 GBP -
Tuberculosis inhibitor 3 [CAS 2219325-28-5]
CAS: 2219325-28-5 | SKU: QM-0138289-01 | Size: 5 mg£301.50 GBP -
TRPV3 antagonist 74a [CAS 1432051-63-2]
CAS: 1432051-63-2 | SKU: QM-0143736-01 | Size: 1 mg£269.91 GBP -
TSHR antagonist S37b [CAS 2143452-22-4]
CAS: 2143452-22-4 | SKU: QM-0143015-01 | Size: 5 mg£551.80 GBP -
TRPV4 agonist-1 (free base) [CAS 2314467-59-7]
CAS: 2314467-59-7 | SKU: QM-0138423-01 | Size: 5 mg£200.66 GBP -
TRPV1 antagonist 3 [CAS 2765294-54-8]
CAS: 2765294-54-8 | SKU: QM-0148260-01 | Size: 5 mg£452.17 GBP -
TSPO ligand-1 [CAS 4560-08-1]
CAS: 4560-08-1 | SKU: QM-0150314-01 | Size: 5 mg£94.75 GBP -
TSPO ligand-2 [CAS 1160640-95-8]
CAS: 1160640-95-8 | SKU: QM-0150316-01 | Size: 5 mg£111.63 GBP -
Tubulin inhibitor 30 [CAS 2873383-67-4]
CAS: 2873383-67-4 | SKU: QM-0150686-01 | Size: 5 mg£301.50 GBP -
Ubiquitin Isopeptidase Inhibitor I, G5 [CAS 108477-18-5]
CAS: 108477-18-5 | SKU: QM-0079638-01 | Size: 5 mg£131.88 GBP -
Tyrosine kinase inhibitor [CAS 1021950-26-4]
CAS: 1021950-26-4 | SKU: QM-0083611-01 | Size: 5 mg£135.25 GBP -
Tubulin inhibitor 6 [CAS 105925-39-1]
CAS: 105925-39-1 | SKU: QM-0145360-01 | Size: 5 mg£94.75 GBP -
Tuberculosis inhibitor 12 [CAS 793729-44-9]
CAS: 793729-44-9 | SKU: QM-0156366-01 | Size: 5 mg£140.88 GBP -
Trypsin Inhibitor, soybean [CAS 9035-81-8]
CAS: 9035-81-8 | SKU: QM-0141863-01 | Size: 50 mg£65.37 GBP -
TRβ agonist 1 [CAS 2770681-85-9]
CAS: 2770681-85-9 | SKU: QM-0067156-01 | Size: 5 mg£1,217.62 GBP -
Tubulin inhibitor 35 [CAS 2247047-77-2]
CAS: 2247047-77-2 | SKU: QM-0071535-01 | Size: 1 mg£145.38 GBP -
Type II topoisomerase inhibitor 1 [CAS 2245691-60-3]
CAS: 2245691-60-3 | SKU: QM-0068774 | Size: 1 Each Price on request -
TrxR inhibitor D9 [CAS 1527513-89-8]
CAS: 1527513-89-8 | SKU: QM-0062968 | Size: 1 Each Price on request -
Tubulin inhibitor 9 [CAS 1151995-69-5]
CAS: 1151995-69-5 | SKU: QM-0146120 | Size: 1 Each Price on request -
Tuberculosis inhibitor 8 [CAS 141353-07-3]
CAS: 141353-07-3 | SKU: QM-0071940 | Size: 1 Each Price on request -
Tubulin inhibitor 26 [CAS 2379241-70-8]
CAS: 2379241-70-8 | SKU: QM-0066808 | Size: 1 Each Price on request -
Tubulin inhibitor 46
SKU: QM-0134344 | Size: 1 Each Price on request -
Tuberculosis inhibitor 1 [CAS 2230810-28-1]
CAS: 2230810-28-1 | SKU: QM-0059741 | Size: 1 Each Price on request -
Tubulin inhibitor 38
SKU: QM-0068334 | Size: 1 Each Price on request -
TTK inhibitor 4 [CAS 2964520-80-5]
CAS: 2964520-80-5 | SKU: QM-0073520 | Size: 1 Each Price on request -
Tubulin inhibitor 24 [CAS 2415761-65-6]
CAS: 2415761-65-6 | SKU: QM-0067052-01 | Size: 1 mg£233.47 GBP -
Tubulin inhibitor 40
SKU: QM-0073694 | Size: 1 Each Price on request -
Tubulin inhibitor 21
SKU: QM-0059162 | Size: 1 Each Price on request -
Tubulin inhibitor 47
SKU: QM-0120795 | Size: 1 Each Price on request -
Type II TRK inhibitor 2
SKU: QM-0073552 | Size: 1 Each Price on request -
TRPV1 antagonist 9 [CAS 939040-79-6]
CAS: 939040-79-6 | SKU: QM-0119839-01 | Size: 500 µg£911.43 GBP -
TRPV4 agonist-1 [CAS 2314467-60-0]
CAS: 2314467-60-0 | SKU: QM-0058919 | Size: 1 Each Price on request -
Tubulin inhibitor 27 [CAS 184579-57-5]
CAS: 184579-57-5 | SKU: QM-0066034 | Size: 1 Each Price on request -
Tubulin inhibitor 19
SKU: QM-0059150 | Size: 1 Each Price on request -
TRβ agonist 3 [CAS 2411099-46-0]
CAS: 2411099-46-0 | SKU: QM-0067337 | Size: 1 Each Price on request